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5,6-Dihydro-3- (4-morpholinyl) -1-[4- (2-oxo-1-piperidinyl) phenyl] -2 (1H) -pyridinone CAS: 545445-44-1

Takaitaccen Bayani:

Lambar Catalog: XD93344
Cas: 545445-44-1
Tsarin kwayoyin halitta: Saukewa: C20H25N3O3
Nauyin Kwayoyin Halitta: 355.43
samuwa: A Stock
Farashin:  
Shiri:  
Kunshin girma: Neman Magana

 


Cikakken Bayani

Tags samfurin

Lambar Catalog XD93344
Sunan samfur 5,6-Dihydro-3- (4-morpholinyl) -1-[4- (2-oxo-1-piperidinyl) phenyl] -2 (1H) -pyridinone
CAS 545445-44-1
Tsarin kwayoyin halittala Saukewa: C20H25N3O3
Nauyin Kwayoyin Halitta 355.43
Bayanin Ajiya yanayi

 

Ƙayyadaddun samfur

Bayyanar Farin foda
Asay 99% min

 

5,6-Dihydro-3- (4-morpholinyl) -1- [4- (2-oxo-1-piperidinyl) phenyl] -2 (1H) -pyridinone, wanda aka fi sani da DMPPHP, wani fili ne na heterocyclic tare da aikace-aikace daban-daban. a cikin ilmin sunadarai na magani da gano magunguna.Anan akwai bayanin amfani da shi a cikin kusan kalmomi 300. DMPHP an san shi don yuwuwarta a matsayin mai ƙarfi da zaɓin hanawa na wasu enzymes da masu karɓa a cikin jikin mutum.Ɗaya daga cikin aikace-aikacen sa na farko shine a fagen hana kinase.Kinases sune enzymes waɗanda ke taka muhimmiyar rawa a cikin hanyoyin siginar tantanin halitta kuma galibi ana haɗa su cikin cututtuka daban-daban, gami da ciwon daji.An gano DMPHP don zaɓin hana takamaiman kinases, ta haka ya katse ɓangarorin sigina waɗanda ke ba da gudummawa ga ci gaban cuta.Wannan ya sa ya zama dan takara mai ban sha'awa don bunkasa hanyoyin da aka yi niyya don cututtuka daban-daban, ciki har da ciwon daji, ƙumburi, da cututtuka na jijiyoyi. Bugu da ƙari, DMPHP ya nuna yiwuwar yin amfani da kayan aiki na anti-inflammatory da immunomodulatory.Kumburi wani martani ne na dabi'a na jiki ga kamuwa da cuta ko rauni amma yana iya zama na dindindin kuma yana haifar da cututtuka daban-daban.DMPPHP ya nuna ikon hana wasu hanyoyin da ake amfani da su, rage samar da masu shiga tsakani.Wannan dukiya ya sa ya zama kayan aiki mai mahimmanci a cikin ci gaba da magungunan ƙwayoyin cuta, yana taimakawa wajen magance cututtuka irin su cututtukan cututtuka na rheumatoid, cututtuka na hanji, da kuma asma.DMPHP kuma an bincikar shi don yiwuwarsa a matsayin wakili na analgesic ko jin zafi. .Jin zafi na yau da kullun shine muhimmin batun kiwon lafiya, kuma zaɓuɓɓukan jiyya na yanzu suna da iyakancewa ko illolin da ba'a so.DMPHP ya nuna alamun analgesic a cikin binciken bincike na yau da kullun, yana ba da shawarar yiwuwarsa a matsayin sabon magani don sarrafa ciwo.Ta hanyar daidaita masu karɓa na musamman da masu amfani da ƙwayoyin cuta da ke cikin jin zafi, DMPPHP na iya ba da wata hanyar da za ta iya ba da wata hanyar da za ta iya magance ciwo mai zafi tare da ƙananan sakamako masu illa. Bugu da ƙari, DMPPHP ya nuna alƙawari a cikin tsarin tsarin juyayi na tsakiya (CNS).Yanayin jijiyoyi kamar cutar Alzheimer da cutar Parkinson sun haɗa da hadaddun ingantattun hanyoyin da dysregulation na daban-daban masu karɓa da enzymes a cikin kwakwalwa.An yi nazarin DMPHP don yuwuwar sa a matsayin wakili na neuroprotective da kuma ikon haɓaka aikin fahimi.Ta hanyar ƙaddamar da ƙayyadaddun masu karɓa da kuma hanyoyin da ke tattare da cututtuka na neurodegenerative, DMPPHP yana riƙe da alkawari a matsayin maganin warkewa don waɗannan yanayi masu kalubale. 1-piperidinyl) phenyl] -2 (1H) -pyridinone (DMPHP) wani nau'i ne mai mahimmanci tare da aikace-aikacen aikace-aikace a cikin hana kinase, aikin anti-inflammatory, analgesia, da neuroprotection.Ƙarfinsa na zaɓin canza takamaiman enzymes da masu karɓa da ke cikin hanyoyin cututtuka ya sa ya zama ɗan takara mai ban sha'awa don gano magunguna da sa baki na warkewa.Ƙarin bincike da haɓakawa na iya buɗe ƙarin amfani da haɓaka kaddarorin sa don takamaiman alamu.


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    5,6-Dihydro-3- (4-morpholinyl) -1-[4- (2-oxo-1-piperidinyl) phenyl] -2 (1H) -pyridinone CAS: 545445-44-1