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Methyl 1-[(2'-cyanobiphenyl-4-yl)methyl]-2-ethoxy-1H-benzimidazole-7-carboxylate CAS: 139481-44-0

Takaitaccen Bayani:

Lambar Catalog: XD93630
Cas: 139481-44-0
Tsarin kwayoyin halitta: Saukewa: C25H21N3O3
Nauyin Kwayoyin Halitta: 411.45
samuwa: A Stock
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Shiri:  
Kunshin girma: Neman Magana

 


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Tags samfurin

Lambar Catalog XD93630
Sunan samfur Methyl 1-[(2'-cyanobiphenyl-4-yl)methyl]-2-ethoxy-1H-benzimidazole-7-carboxylate
CAS 139481-44-0
Tsarin kwayoyin halittala Saukewa: C25H21N3O3
Nauyin Kwayoyin Halitta 411.45
Bayanin Ajiya yanayi

Ƙayyadaddun samfur

Bayyanar Farin foda
Asay 99% min

 

Methyl 1- [(2'-cyanobiphenyl-4-yl) methyl] -2-ethoxy-1H-benzimidazole-7-carboxylate wani sinadari ne mai amfani da yuwuwar amfani a aikace-aikace daban-daban, da farko a fagen magunguna. dangin benzimidazole, waɗanda aka bincika ko'ina don yuwuwar warkewar su.An gano Benzimidazoles don nuna nau'o'in ayyukan ilimin halitta, ciki har da anticancer, antifungal, antibacterial, antiviral, da anti-inflammatory Properties.Methyl 1-[(2'-cyanobiphenyl-4-yl) methyl] -2-ethoxy-1H -benzimidazole-7-carboxylate na iya aiki a matsayin sifa ko ginshiƙan tsari don ƙira da haɓaka sabbin ƙwayoyi.Tsarin sinadarai na musamman yana ba da dama don ƙarin gyare-gyare da haɓakawa don haɓaka ayyukan harhada magunguna da ake so ko manufa takamaiman hanyoyin cuta.Masanan ilimin likitanci na iya amfani da wannan fili a matsayin mafari don haɗa sabbin kwayoyin halitta tare da yuwuwar aikace-aikacen warkewa.Ta hanyar gabatar da abubuwan maye gurbin sinadarai masu dacewa ko ƙungiyoyi masu aiki akan ainihin tsarin, masu bincike na iya ƙirƙirar abubuwan da suka mallaki ingantaccen ƙarfi, zaɓi, da kaddarorin pharmacokinetic.Wadannan gyare-gyare na iya haɓaka tasirin mahallin a cikin ƙaddamar da ƙayyadaddun hanyoyin cututtuka ko maƙasudin kwayoyin halitta, wanda zai haifar da haɓakar magunguna masu mahimmanci.Za'a iya gudanar da gwaje-gwaje da nazari don kimanta ayyukan nazarin halittu na fili ta hanyar amfani da in vitro cell-based assays ko a cikin samfurin dabba na vivo.Wannan zai iya ba da haske mai mahimmanci game da yiwuwar aikace-aikacen warkewa da kuma jagorantar ƙarin haɓakawa. Bugu da ƙari, wannan fili zai iya zama kayan aiki mai mahimmanci a cikin nazarin tsarin-aikin dangantaka (SAR) na benzimidazole.Ta hanyar haɗa analogs tare da bambance-bambance a cikin sarƙoƙi na gefe ko ƙungiyoyin aiki, masana kimiyya za su iya samun kyakkyawar fahimtar yadda takamaiman gyare-gyaren tsarin ke shafar ayyukan fili da zaɓin.Wannan ilimin zai iya taimakawa wajen tsara ma'auni na 'yan takarar magunguna masu mahimmanci da zaɓaɓɓu.Bugu da ƙari, wannan fili na iya yiwuwa a yi amfani da shi a cikin ci gaban prodrugs, inda za a iya zabar rukunin ethoxy, yana sakin miyagun ƙwayoyi mai aiki a wurin da aka yi niyya.Prodrugs suna ba da fa'idodi kamar ingantaccen solubility, haɓakar haɓakar haɓakar rayuwa, da isar da takamaiman nama, ta haka inganta tasirin miyagun ƙwayoyi da rage tasirin sakamako.Duk da haka, yana da mahimmanci a lura cewa ƙarin bincike, ingantaccen kimantawa na ƙima, da tsauraran aminci da binciken guba ya zama dole. kafin yin la'akari da fili don ci gaban asibiti.Wannan yana da mahimmanci don tabbatar da amincinsa, inganci, da dacewa don aikace-aikacen warkewa.A ƙarshe, Methyl 1-[(2'-cyanobiphenyl-4-yl) methyl]-2-ethoxy-1H-benzimidazole-7-carboxylate yana ɗaukar alkawari kamar wani m fili tare da m aikace-aikace a fagen Pharmaceuticals.Tsarinsa na musamman da kaddarorin sinadarai suna ba da damammaki don gano magunguna, haɓakawa, da haɓaka samfuran magunguna.Koyaya, ana buƙatar ƙarin bincike da gwaji don cikakken bincika yuwuwar warkewarsa da tabbatar da amincin sa don amfanin asibiti.


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    Methyl 1-[(2'-cyanobiphenyl-4-yl)methyl]-2-ethoxy-1H-benzimidazole-7-carboxylate CAS: 139481-44-0